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CCc1cc2c(cc1N1CCC(N(C)Cc3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC1)C(C)(C)c1[nH]c3cc(C#N)ccc3c1C2=O| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | ALK | - | SR | CN116239566A | PGDB_A022255 | PGDB_C019614 | PGDB_AS001815 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | ALK | - | MDA-MB-231 | CN116239566A | PGDB_A031129 | PGDB_C019614 | PGDB_AS000594 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | ALK | - | HCC827 | CN116239566A | PGDB_A032516 | PGDB_C019614 | PGDB_AS000527 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | ALK | - | PC-9 | CN116239566A | PGDB_A052095 | PGDB_C019614 | PGDB_AS000139 | View |