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O=C1CCC(N2Cc3cc(CN4CCC(N(c5ccccc5)c5ccccc5)CC4)ccc3C2=S)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 80-100 | % | - | - | - | - | - | CN119654316A | PGDB_A082114 | PGDB_C022011 | PGDB_AS000466 | View | |
| IC50 | - | > | 10 | nM | - | — | - | - | MCF-7 | CN119654316A | PGDB_A082206 | PGDB_C022011 | PGDB_AS001496 | View | |
| IC50 | - | > | 0 | nM | - | — | - | - | MM.1S | CN119654316A | PGDB_A082373 | PGDB_C022011 | PGDB_AS001506 | View | |
| % Degradation | - | = | 0-80 | % | - | - | IKZF2 | - | - | CN119654316A | PGDB_A082501 | PGDB_C022011 | PGDB_AS002430 | View | |
| IC50 | - | > | 0 | nM | - | — | - | - | Jurkat | CN119654316A | PGDB_A082776 | PGDB_C022011 | PGDB_AS002479 | View | |
| % Degradation | - | = | 0-80 | % | - | - | GSPT1 | - | - | CN119654316A | PGDB_A082924 | PGDB_C022011 | PGDB_AS000660 | View | |
| % Degradation | - | = | 0-80 | % | - | - | IKZF3 | - | - | CN119654316A | PGDB_A083383 | PGDB_C022011 | PGDB_AS000017 | View | |
| IC50 | - | > | 5 | nM | - | — | - | - | MGC-803 | CN119654316A | PGDB_A083809 | PGDB_C022011 | PGDB_AS002336 | View | |
| % Degradation | - | = | 0-80 | % | - | - | WEE1 | - | - | CN119654316A | PGDB_A083869 | PGDB_C022011 | PGDB_AS001023 | View | |
| IC50 | - | > | 0 | nM | - | — | - | - | JeKo-1 | CN119654316A | PGDB_A084575 | PGDB_C022011 | PGDB_AS000137 | View | |
| IC50 | - | > | 5 | nM | - | — | - | - | H1975 | CN119654316A | PGDB_A084908 | PGDB_C022011 | PGDB_AS002346 | View | |
| % Degradation | - | = | 0-80 | % | - | - | IKZF1 | - | - | CN119654316A | PGDB_A085060 | PGDB_C022011 | PGDB_AS001680 | View |