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Cc1ccc(C2=CCN(Cc3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=S)CC2)s1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | > | 100 | nM | - | — | - | - | MCF-7 | CN119654316A | PGDB_A082223 | PGDB_C022013 | PGDB_AS001496 | View | |
| IC50 | - | > | 50 | nM | - | — | - | - | H1975 | CN119654316A | PGDB_A083192 | PGDB_C022013 | PGDB_AS002346 | View | |
| % Degradation | - | = | 0-80 | % | - | - | GSPT1 | - | - | CN119654316A | PGDB_A083815 | PGDB_C022013 | PGDB_AS000660 | View | |
| IC50 | - | > | 50 | nM | - | — | - | - | Jurkat | CN119654316A | PGDB_A083989 | PGDB_C022013 | PGDB_AS002479 | View | |
| % Degradation | - | = | 0-80 | % | - | - | IKZF1 | - | - | CN119654316A | PGDB_A084102 | PGDB_C022013 | PGDB_AS001680 | View | |
| % Degradation | - | = | 0-80 | % | - | - | WEE1 | - | - | CN119654316A | PGDB_A084211 | PGDB_C022013 | PGDB_AS001023 | View | |
| IC50 | - | > | 10 | nM | - | — | - | - | MM.1S | CN119654316A | PGDB_A084414 | PGDB_C022013 | PGDB_AS001506 | View | |
| % Degradation | - | = | 0-80 | % | - | - | - | - | - | CN119654316A | PGDB_A084483 | PGDB_C022013 | PGDB_AS000466 | View | |
| IC50 | - | > | 100 | nM | - | — | - | - | MGC-803 | CN119654316A | PGDB_A084695 | PGDB_C022013 | PGDB_AS002336 | View | |
| IC50 | - | > | 50 | nM | - | — | - | - | JeKo-1 | CN119654316A | PGDB_A085027 | PGDB_C022013 | PGDB_AS000137 | View | |
| % Degradation | - | = | 0-80 | % | - | - | IKZF2 | - | - | CN119654316A | PGDB_A085149 | PGDB_C022013 | PGDB_AS002430 | View | |
| % Degradation | - | = | 0-80 | % | - | - | IKZF3 | - | - | CN119654316A | PGDB_A085259 | PGDB_C022013 | PGDB_AS000017 | View |