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Compound
PGDB_C024656
3 activity records1 related patents
2D structure
CCn1c(-c2cc(C#CC(C)(C)C(=O)N3CCN(C)CC3)cnc2C(C)OC)c2c3cc(ccc31)N1CCO[C@@H](C[C@H](NC(=O)[C@H](C(C)C)N3CC[C@]4(CCN(C(=O)[C@H]5[C@@H]6CC6CN5C)C4)C3)C(=O)N3CCC[C@H](N3)C(=O)NCC(C)(C)C2)C1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 10-100 | nM | - | — | KRAS | - | HPAC | CN121181579A | PGDB_A012906 | PGDB_C024656 | PGDB_AS000097 | View |
| IC50 | - | <= | 10 | nM | - | — | KRAS | - | AGS | CN121181579A | PGDB_A028109 | PGDB_C024656 | PGDB_AS000586 | View |
| IC50 | - | <= | 10 | nM | - | — | KRAS | - | AsPC-1 | CN121181579A | PGDB_A060179 | PGDB_C024656 | PGDB_AS001095 | View |