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COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1OCc1ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=O| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 1000-5000 | nM | - | — | EGFR | - | NCI-H358 | CN116239566A | PGDB_A016405 | PGDB_C025848 | PGDB_AS000770 | View | |
| IC50 | - | < | 50 | nM | - | — | EGFR | - | HCC827 | CN116239566A | PGDB_A073876 | PGDB_C025848 | PGDB_AS002229 | View |