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COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NCc1ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=O| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 50-100 | nM | - | — | EGFR | - | HCC827 | CN116239566A | PGDB_A026498 | PGDB_C025850 | PGDB_AS002229 | View | |
| IC50 | - | = | 100-500 | nM | - | — | EGFR | - | PC-9 | CN116239566A | PGDB_A032928 | PGDB_C025850 | PGDB_AS000044 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | EGFR | - | NCI-H358 | CN116239566A | PGDB_A066267 | PGDB_C025850 | PGDB_AS000770 | View |