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CN(Cc1ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=O)C1CCN(c2ccc(Nc3ncc4nc(Nc5ccccc5)n(C5CCCC5)c4n3)cc2)CC1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 50-100 | nM | - | — | EGFR | - | Mino | CN116239566A | PGDB_A019775 | PGDB_C025855 | PGDB_AS000353 | View | |
| IC50 | - | = | 50-100 | nM | - | — | EGFR | - | Mino | CN116239566A | PGDB_A043561 | PGDB_C025855 | PGDB_AS000353 | View | |
| IC50 | - | = | 100-500 | nM | - | — | EGFR | - | SR | CN116239566A | PGDB_A043994 | PGDB_C025855 | PGDB_AS001321 | View | |
| IC50 | - | < | 50 | nM | - | — | EGFR | - | THP-1 | CN116239566A | PGDB_A068775 | PGDB_C025855 | PGDB_AS002327 | View | |
| IC50 | - | < | 50 | nM | - | — | EGFR | - | PC-9 | CN116239566A | PGDB_A068973 | PGDB_C025855 | PGDB_AS000044 | View | |
| IC50 | - | < | 50 | nM | - | — | EGFR | - | PC-9 | CN116239566A | PGDB_A071212 | PGDB_C025855 | PGDB_AS000044 | View |