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O=C1CCC(N2Cc3cc(CN4CCC(N5CCN(c6ccc(-c7cc(F)c8c(c7)C(=O)N(C(C(=O)Nc7nccs7)c7ncn9c7CCC9)C8)cc6)CC5)C(F)(F)C4)ccc3C2=O)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | EGFR | - | VCaP | CN116239566A | PGDB_A013034 | PGDB_C025856 | PGDB_AS001793 | View | |
| IC50 | - | < | 50 | nM | - | — | EGFR | - | CCRF-CEM | CN116239566A | PGDB_A015113 | PGDB_C025856 | PGDB_AS000005 | View | |
| IC50 | - | = | 50-100 | nM | - | — | EGFR | - | SR | CN116239566A | PGDB_A030166 | PGDB_C025856 | PGDB_AS001321 | View | |
| IC50 | - | < | 50 | nM | - | — | EGFR | - | THP-1 | CN116239566A | PGDB_A041828 | PGDB_C025856 | PGDB_AS002327 | View |