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COc1cc(Nc2c(C#N)cnc3cc(OCCCN4CCN(Cc5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)c(OC)cc23)c(Cl)cc1Cl| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 1000-5000 | nM | - | — | ABL1 | - | Kasumi-1 | CN116239566A | PGDB_A025851 | PGDB_C025885 | PGDB_AS000069 | View | |
| IC50 | - | = | 50-100 | nM | - | — | ABL1 | - | K562 | CN116239566A | PGDB_A034498 | PGDB_C025885 | PGDB_AS002026 | View | |
| IC50 | - | < | 50 | nM | - | — | ABL1 | - | CCRF-CEM | CN116239566A | PGDB_A054582 | PGDB_C025885 | PGDB_AS000919 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | ABL1 | - | Daudi | CN116239566A | PGDB_A067907 | PGDB_C025885 | PGDB_AS001018 | View |