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Cc1ccc(C(=O)Nc2ccc(N3CCN(Cc4ccc5c(c4)CN(C4CCC(=O)NC4=O)C5=O)CC3)c(C(F)(F)F)c2)cc1C#Cc1cnc2cccnn12| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | ABL1 | - | K562 | CN116239566A | PGDB_A008498 | PGDB_C025890 | PGDB_AS002026 | View | |
| IC50 | - | < | 50 | nM | - | — | ABL1 | - | CCRF-CEM | CN116239566A | PGDB_A014098 | PGDB_C025890 | PGDB_AS000919 | View | |
| IC50 | - | = | 100-500 | nM | - | — | ABL1 | - | Kasumi-1 | CN116239566A | PGDB_A039562 | PGDB_C025890 | PGDB_AS000069 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | ABL1 | - | CAL-62 | CN116239566A | PGDB_A057544 | PGDB_C025890 | PGDB_AS000882 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | ABL1 | - | Daudi | CN116239566A | PGDB_A067877 | PGDB_C025890 | PGDB_AS001018 | View |