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CC(C)Nc1cc(-n2ccc3cc(C#N)cnc32)ncc1C(=O)N[C@H]1CC[C@H](C(=O)NCc2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)CC1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | SW620 | CN116239566A | PGDB_A019728 | PGDB_C025975 | PGDB_AS000233 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | LNCaP | CN116239566A | PGDB_A023222 | PGDB_C025975 | PGDB_AS000964 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | SU-DHL-4 | CN116239566A | PGDB_A038152 | PGDB_C025975 | PGDB_AS002569 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | CAL-62 | CN116239566A | PGDB_A043785 | PGDB_C025975 | PGDB_AS000175 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | Jurkat | CN116239566A | PGDB_A063981 | PGDB_C025975 | PGDB_AS000478 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | CCRF-CEM | CN116239566A | PGDB_A064052 | PGDB_C025975 | PGDB_AS001036 | View |