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CO[C@@H](C)c1ncc(C#CCN2CC[C@@H](F)C2)cc1-c1c2c3cc(cc4c3n1CCO4)-c1csc(n1)C[C@H](CC(=O)[C@H]1[C@H](C)[C@@H]1C)NC(=O)C1C[C@@H](N1)C(=O)OCC(C)(C)C2| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | > | 1 | nM | - | — | KRAS | - | HPAC | WO2026047641A1 | PGDB_A007147 | PGDB_C028435 | PGDB_AS001191 | View | |
| IC50 | - | > | 1 | nM | - | — | KRAS | - | SW620 | WO2026047641A1 | PGDB_A030202 | PGDB_C028435 | PGDB_AS000598 | View | |
| IC50 | - | > | 1 | nM | - | — | KRAS | - | NCI-H358 | WO2026047641A1 | PGDB_A037753 | PGDB_C028435 | PGDB_AS001839 | View | |
| IC50 | - | > | 1 | nM | - | — | KRAS | - | AGS | WO2026047641A1 | PGDB_A041253 | PGDB_C028435 | PGDB_AS000159 | View | |
| IC50 | - | > | 1 | nM | - | — | KRAS | - | AsPC-1 | WO2026047641A1 | PGDB_A041727 | PGDB_C028435 | PGDB_AS000949 | View |