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Compound
PGDB_C028700
5 activity records1 related patents
2D structure
Cc1nn(CC(=O)Nc2ccc3c(F)c(N4CC(=O)NS4(=O)=O)c4[nH]ncc4c3c2)c(C)c1-c1ccc2c(C3CCC(=O)NC3=O)nn(C)c2c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 97.6 | % | - | - | - | - | - | WO2026119184 | PGDB_A026852 | PGDB_C028700 | PGDB_AS001850 | View |
| DC50 | - | = | 15.64 | nM | - | — | - | - | - | WO2026119184 | PGDB_A036377 | PGDB_C028700 | PGDB_AS002400 | View |
| DC50 | - | = | 15.25 | nM | - | — | PTPN1 | - | - | WO2026119184 | PGDB_A039523 | PGDB_C028700 | PGDB_AS000433 | View |
| Selectivity index | N2/1B | = | 0.98 | fold | - | — | - | - | - | WO2026119184 | PGDB_A060385 | PGDB_C028700 | PGDB_AS001537 | View |
| Dmax | - | = | 93.7 | % | - | - | PTPN1 | - | - | WO2026119184 | PGDB_A065762 | PGDB_C028700 | PGDB_AS002412 | View |