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Nc1nnc(-c2cc(F)ccc2O)cc1N1CC2CCC(C1)N2c1cccc(CN2CCN(Cc3ccc(N4CCC(=O)NC4=O)cc3)CC2)c1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 100-200 | nM | - | — | - | - | H838 | WO2026061475A1 | PGDB_A000190 | PGDB_C030312 | PGDB_AS000282 | View | |
| IC50 | - | = | 700-900 | nM | - | — | - | - | BT549 | WO2026061475A1 | PGDB_A001672 | PGDB_C030312 | PGDB_AS002259 | View | |
| IC50 | - | = | 700-900 | nM | - | — | - | - | A549 | WO2026061475A1 | PGDB_A004218 | PGDB_C030312 | PGDB_AS000757 | View | |
| IC50 | - | = | 50-100 | nM | - | — | - | - | H1944 | WO2026061475A1 | PGDB_A005382 | PGDB_C030312 | PGDB_AS001924 | View | |
| IC50 | - | = | 10-20 | nM | - | — | - | - | H2126 | WO2026061475A1 | PGDB_A081111 | PGDB_C030312 | PGDB_AS001417 | View |