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Compound
PGDB_C030317
9 activity records1 related patents
2D structure
Nc1nnc(-c2cc(F)ccc2O)cc1N1CC2CCC(C1)N2c1cccc(CN2CCN(Cc3cccc(NC4CCC(=O)NC4=O)c3)CC2)c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 50-100 | nM | - | — | - | - | H2126 | WO2026061475A1 | PGDB_A002661 | PGDB_C030317 | PGDB_AS001417 | View |
| IC50 | - | = | 200-500 | nM | - | — | - | - | H838 | WO2026061475A1 | PGDB_A003762 | PGDB_C030317 | PGDB_AS000282 | View |
| IC50 | - | = | 100-200 | nM | - | — | - | - | A549 | WO2026061475A1 | PGDB_A005844 | PGDB_C030317 | PGDB_AS000757 | View |
| % Degradation | - | <= | 50 | % | Concentration series: 500 nM, 50 nM | - | SMARCA2 | - | MV-4-11 | WO2026061475A1 | PGDB_A080107 | PGDB_C030317 | PGDB_AS002335 | View |
| IC50 | - | = | 100-200 | nM | - | — | - | - | H1944 | WO2026061475A1 | PGDB_A080677 | PGDB_C030317 | PGDB_AS001924 | View |