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SIMM · NJU
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SIMM · NJU
Patent
CN112566886A
15 compounds
15 activity records
1 assays
Patent summary
Publication number
CN112566886A
Assignee
C4 Therapeutics
Title
Spiro compounds
Family ID
62528307
Family members
9
Family patent IDs
CN112566886A
CN119751465A
EP3578561A1
EP3802467A1
EP3802467A4
US11623929B2
US20210070763A1
US20240018156A1
WO2019236483A1
Filing year
2019
Publication date
2021-03-26
Jurisdiction
CN
Compounds
15
Activity records
15
Assays
1
Activity compounds and values
Activity records
15 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Record ID
Compound
Assay
Details
Kd
-
=
0.018
uM
-
—
CRBN
CRBN
-
PGDB_A009465
PGDB_C006467
PGDB_AS000393
View
Kd
-
=
0.032
uM
-
—
CRBN
CRBN
-
PGDB_A019969
PGDB_C006465
PGDB_AS000393
View
Kd
-
=
0.01
uM
-
—
CRBN
CRBN
-
PGDB_A028783
PGDB_C006462
PGDB_AS000393
View
Kd
-
=
0.037
uM
-
—
CRBN
CRBN
-
PGDB_A035316
PGDB_C006460
PGDB_AS000393
View
Kd
-
=
0.026
uM
-
—
CRBN
CRBN
-
PGDB_A040192
PGDB_C026001
PGDB_AS000393
View
Kd
-
=
0.002
uM
-
—
CRBN
CRBN
-
PGDB_A044897
PGDB_C006461
PGDB_AS000393
View
Kd
-
=
0.003
uM
-
—
CRBN
CRBN
-
PGDB_A046058
PGDB_C006458
PGDB_AS000393
View
Kd
-
=
0.007
uM
-
—
CRBN
CRBN
-
PGDB_A048845
PGDB_C006464
PGDB_AS000393
View
Kd
-
=
0.015
uM
-
—
CRBN
CRBN
-
PGDB_A050265
PGDB_C006469
PGDB_AS000393
View
Kd
-
=
0.006
uM
-
—
CRBN
CRBN
-
PGDB_A050939
PGDB_C025999
PGDB_AS000393
View
Kd
-
=
0.004
uM
-
—
CRBN
CRBN
-
PGDB_A052441
PGDB_C006457
PGDB_AS000393
View
Kd
-
=
0.01
uM
-
—
CRBN
CRBN
-
PGDB_A064292
PGDB_C006466
PGDB_AS000393
View
Kd
-
=
0.031
uM
-
—
CRBN
CRBN
-
PGDB_A065459
PGDB_C006459
PGDB_AS000393
View
Kd
-
=
0.023
uM
-
—
CRBN
CRBN
-
PGDB_A068045
PGDB_C011110
PGDB_AS000393
View
Kd
-
=
0.161
uM
-
—
CRBN
CRBN
-
PGDB_A069862
PGDB_C006463
PGDB_AS000393
View