Assay

PGDB_AS000393

System: biochemicalTarget: CRBN | DDB1
Assay context summary

Assay context

15 activity records
Assay familybinding
Systembiochemical
ReadoutKd
TargetCRBN | DDB1
E3CRBN | DDB1
OrganismHomo sapiens
Technologyfluorescence
Activity compounds and values

Activity records

15 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C006467
Kd-=0.018uM-—CRBNCRBN-CN112566886APGDB_A009465PGDB_C006467PGDB_AS000393View
2D structure for PGDB_C006465
Kd-=0.032uM-—CRBNCRBN-CN112566886APGDB_A019969PGDB_C006465PGDB_AS000393View
2D structure for PGDB_C006462
Kd-=0.01uM-—CRBNCRBN-CN112566886APGDB_A028783PGDB_C006462PGDB_AS000393View
2D structure for PGDB_C006460
Kd-=0.037uM-—CRBNCRBN-CN112566886APGDB_A035316PGDB_C006460PGDB_AS000393View
2D structure for PGDB_C026001
Kd-=0.026uM-—CRBNCRBN-CN112566886APGDB_A040192PGDB_C026001PGDB_AS000393View
2D structure for PGDB_C006461
Kd-=0.002uM-—CRBNCRBN-CN112566886APGDB_A044897PGDB_C006461PGDB_AS000393View
2D structure for PGDB_C006458
Kd-=0.003uM-—CRBNCRBN-CN112566886APGDB_A046058PGDB_C006458PGDB_AS000393View
2D structure for PGDB_C006464
Kd-=0.007uM-—CRBNCRBN-CN112566886APGDB_A048845PGDB_C006464PGDB_AS000393View
2D structure for PGDB_C006469
Kd-=0.015uM-—CRBNCRBN-CN112566886APGDB_A050265PGDB_C006469PGDB_AS000393View
2D structure for PGDB_C025999
Kd-=0.006uM-—CRBNCRBN-CN112566886APGDB_A050939PGDB_C025999PGDB_AS000393View
2D structure for PGDB_C006457
Kd-=0.004uM-—CRBNCRBN-CN112566886APGDB_A052441PGDB_C006457PGDB_AS000393View
2D structure for PGDB_C006466
Kd-=0.01uM-—CRBNCRBN-CN112566886APGDB_A064292PGDB_C006466PGDB_AS000393View
2D structure for PGDB_C006459
Kd-=0.031uM-—CRBNCRBN-CN112566886APGDB_A065459PGDB_C006459PGDB_AS000393View
2D structure for PGDB_C011110
Kd-=0.023uM-—CRBNCRBN-CN112566886APGDB_A068045PGDB_C011110PGDB_AS000393View
2D structure for PGDB_C006463
Kd-=0.161uM-—CRBNCRBN-CN112566886APGDB_A069862PGDB_C006463PGDB_AS000393View
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