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Patent
RU2847441C1
4 compounds16 activity records4 assays
Patent summary
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | ||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
 | % Cell viability | - | = | 13 | % | Concentration range: 10 uM | 5 d | ESR1 | - | MCF-7 | PGDB_A009831 | PGDB_C008967 | PGDB_AS002582 | View |
 | IC50 | - | = | 0.07 | nM | - | — | ESR1 | - | MCF-7 | PGDB_A013222 | PGDB_C008966 | PGDB_AS001905 | View |
 | IC50 | - | = | 0.2 | nM | - | — | ESR1 | - | MCF-7 | PGDB_A021288 | PGDB_C008964 | PGDB_AS002097 | View |
 | % Degradation | - | = | 97 | % | Concentration context: 5.12x10⁻¹² M, 5.12x10⁻¹³ M | 4 h | ESR1 | - | MCF-7 | PGDB_A025453 | PGDB_C008965 | PGDB_AS002178 | View |
| IC50 | - | = | 0.05 | nM | - | — | ESR1 | - | MCF-7 | PGDB_A025684 | PGDB_C008966 | PGDB_AS002097 | View |
| IC50 | - | = | 0.21 | nM | - | — | ESR1 | - | MCF-7 | PGDB_A025938 | PGDB_C008964 | PGDB_AS001905 | View |
| IC50 | - | = | 0.3 | nM | - | — | ESR1 | - | MCF-7 | PGDB_A035799 | PGDB_C008967 | PGDB_AS002097 | View |
| % Cell viability | - | = | 4 | % | Concentration range: 10 uM | 5 d | ESR1 | - | MCF-7 | PGDB_A041576 | PGDB_C008964 | PGDB_AS002582 | View |
| % Degradation | - | = | 97 | % | Concentration context: 5.12x10⁻¹² M, 5.12x10⁻¹³ M | 4 h | ESR1 | - | MCF-7 | PGDB_A041961 | PGDB_C008964 | PGDB_AS002178 | View |
| % Cell viability | - | = | 4 | % | Concentration range: 10 uM | 5 d | ESR1 | - | MCF-7 | PGDB_A042245 | PGDB_C008965 | PGDB_AS002582 | View |
| IC50 | - | = | 4.3 | nM | - | — | ESR1 | - | MCF-7 | PGDB_A042549 | PGDB_C008965 | PGDB_AS001905 | View |
| % Degradation | - | = | 97 | % | Concentration context: 5.12x10⁻¹² M, 5.12x10⁻¹³ M | 4 h | ESR1 | - | MCF-7 | PGDB_A049738 | PGDB_C008966 | PGDB_AS002178 | View |
| % Cell viability | - | = | 2 | % | Concentration range: 10 uM | 5 d | ESR1 | - | MCF-7 | PGDB_A050885 | PGDB_C008966 | PGDB_AS002582 | View |
| IC50 | - | = | 0.2 | nM | - | — | ESR1 | - | MCF-7 | PGDB_A057747 | PGDB_C008967 | PGDB_AS001905 | View |
| % Degradation | - | = | 86 | % | Concentration context: 5.12x10⁻¹² M, 5.12x10⁻¹³ M | 4 h | ESR1 | - | MCF-7 | PGDB_A068547 | PGDB_C008967 | PGDB_AS002178 | View |
| IC50 | - | = | 3.4 | nM | - | — | ESR1 | - | MCF-7 | PGDB_A077179 | PGDB_C008965 | PGDB_AS002097 | View |