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SIMM · NJU
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SIMM · NJU
Patent
WO2026114368A1
73 compounds
244 activity records
4 assays
Patent summary
Publication number
WO2026114368A1
Assignee
Xizang Haisco Pharmaceutical Co Ltd
Title
VAV1-TARGETING DEGRADER AND USE THEREOF
Family ID
unresolved_family_WO2026114368A1
Family members
1
Family patent IDs
WO2026114368A1
Filing year
2025
Publication date
2026-06-04
Jurisdiction
WO
Compounds
73
Activity records
244
Assays
4
Activity compounds and values
Activity records
116 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Record ID
Compound
Assay
Details
DC50
-
<=
20
nM
-
—
VAV1
-
-
PGDB_A000051
PGDB_C031883
PGDB_AS000780
View
IC50
-
<=
1
nM
-
—
VAV1
-
primaryT
PGDB_A000090
PGDB_C031870
PGDB_AS001463
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
PGDB_A000100
PGDB_C031873
PGDB_AS000780
View
IC50
-
<=
1
nM
-
—
VAV1
-
primaryT
PGDB_A000404
PGDB_C031865
PGDB_AS001463
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
PGDB_A000949
PGDB_C031899
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
PGDB_A001015
PGDB_C031925
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
PGDB_A001286
PGDB_C031936
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
PGDB_A001519
PGDB_C031865
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
PGDB_A001691
PGDB_C031887
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
PGDB_A001721
PGDB_C031883
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
PGDB_A001877
PGDB_C031912
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
PGDB_A001892
PGDB_C031903
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
PGDB_A001913
PGDB_C031889
PGDB_AS000052
View
IC50
-
<=
1
nM
-
—
VAV1
-
primaryT
PGDB_A001956
PGDB_C031867
PGDB_AS000300
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
PGDB_A002018
PGDB_C031893
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
PGDB_A002063
PGDB_C031877
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
PGDB_A002106
PGDB_C031881
PGDB_AS000780
View
IC50
-
<=
1
nM
-
—
VAV1
-
primaryT
PGDB_A002129
PGDB_C031869
PGDB_AS001463
View
IC50
-
<=
1
nM
-
—
VAV1
-
primaryT
PGDB_A002230
PGDB_C031870
PGDB_AS000300
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
PGDB_A002237
PGDB_C031916
PGDB_AS000052
View