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SIMM · NJU
Assay
PGDB_AS000780
System: cell_based
Target: VAV1
Assay context summary
Assay context
51 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
VAV1
E3
Not specified
Organism
Homo sapiens
Technology
flow_cytometry
Detection target
protein_degradation
Activity compounds and values
Activity records
51 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A000051
PGDB_C031883
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A000100
PGDB_C031873
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A000949
PGDB_C031899
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A001286
PGDB_C031936
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A001877
PGDB_C031912
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A002063
PGDB_C031877
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A002106
PGDB_C031881
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A002432
PGDB_C031923
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A002646
PGDB_C031865
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A003318
PGDB_C031895
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A003542
PGDB_C031892
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A003553
PGDB_C031928
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A003911
PGDB_C031925
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A004133
PGDB_C031900
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A004257
PGDB_C031897
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A004280
PGDB_C031866
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A004645
PGDB_C031935
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A004698
PGDB_C031924
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A004733
PGDB_C031870
PGDB_AS000780
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A005296
PGDB_C031917
PGDB_AS000780
View