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SIMM · NJU
Assay
PGDB_AS000052
System: cell_based
Target: VAV1
Assay context summary
Assay context
51 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
VAV1
E3
Not specified
Organism
Homo sapiens
Technology
flow_cytometry
Detection target
protein_degradation
Activity compounds and values
Activity records
51 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A001015
PGDB_C031925
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A001519
PGDB_C031865
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A001691
PGDB_C031887
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A001721
PGDB_C031883
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A001892
PGDB_C031903
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A001913
PGDB_C031889
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A002018
PGDB_C031893
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A002237
PGDB_C031916
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A002767
PGDB_C031917
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A002845
PGDB_C031881
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A003263
PGDB_C031877
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A003368
PGDB_C031908
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A003501
PGDB_C031891
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A003590
PGDB_C031912
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A003722
PGDB_C031876
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A004098
PGDB_C031907
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A004117
PGDB_C031928
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A004373
PGDB_C031901
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A004656
PGDB_C031896
PGDB_AS000052
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114368A1
PGDB_A004727
PGDB_C031895
PGDB_AS000052
View