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SIMM · NJU
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·
SIMM · NJU
Target
GSPT1
8,970 activity records
5,504 compounds
79 patents
Target summary
Target ID
PGDB_T000034
Name
GSPT1
Gene symbol
GSPT1
Protein name
Eukaryotic peptide chain release factor GTP-binding subunit ERF3A
UniProt ID
P15170
Role
assay_context_marker | assay_marker | degradation_target | effector | neo_substrate | primary_target
Compounds
5,504
Activity records
8,970
Assays
207
Patents
79
Activity compounds and values
Activity records
8,970 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A000098
PGDB_C031976
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A000359
PGDB_C031995
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A000467
PGDB_C031943
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A000626
PGDB_C031993
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A000705
PGDB_C031984
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A000860
PGDB_C031946
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A001013
PGDB_C031976
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A001207
PGDB_C031989
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A001506
PGDB_C031973
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A001509
PGDB_C031959
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A001559
PGDB_C031974
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A001711
PGDB_C031954
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A002037
PGDB_C031975
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A002153
PGDB_C031953
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A002506
PGDB_C031968
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A002530
PGDB_C031988
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A002599
PGDB_C031952
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A002687
PGDB_C031969
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A002773
PGDB_C031950
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A003210
PGDB_C031964
PGDB_AS001690
View