Activity record

PGDB_A008880

Assay: viabilityTarget: GSPT1QC: standardized
Activity overview

IC50 = 3.7 nM

TargetGSPT1
Cell lineMOLM-13
TimeThree days later
Assay / ReadoutIC50 / viability
Assay IDPGDB_AS001125
PatentWO2022073469A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C004695
Compound IDPGDB_C004695
CompoundGS-060;GS-060
Source record IDPGDB_C004695
InChIKeyWPQADJBPJPOUQI-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001125
Assay familyviability
Assay systemcell_based
ReadoutIC50
Treatment timeThree days later
Detection target% Cell viability
TargetGSPT1
E3Not specified
Cell lineMOLM-13

Source evidence

Patent IDWO2022073469A1
Compound location

GS-060;GS-060

GS-060;GS-060 enlarged structureGS-060;GS-060 location on patent page 179
Activity table
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