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O=C1CCC(N2C(=O)c3ccc(NCCCCCC(=O)N4CCC(c5cnc6cccc(Br)c6n5)CC4)cc3C2=O)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 3.7 | nM | - | — | GSPT1 | - | MOLM-13 | WO2022073469A1 | PGDB_A008880 | PGDB_C004695 | PGDB_AS001125 | View | |
| IC50 | - | = | 0.06 | nM | - | — | GSPT1 | - | MOLM-13 | WO2022073469A1 | PGDB_A021744 | PGDB_C004695 | PGDB_AS001795 | View | |
| IC50 | - | < | 10 | nM | - | — | GSPT1 | - | MOLM-13 | WO2022073469A1 | PGDB_A047610 | PGDB_C004695 | PGDB_AS000952 | View | |
| IC50 | - | < | 10 | nM | - | — | - | - | MV-4-11 | WO2022073469A1 | PGDB_A049099 | PGDB_C004695 | PGDB_AS000609 | View | |
| IC50 | - | < | 10 | nM | - | — | GSPT1 | - | MOLM-13 | WO2022073469A1 | PGDB_A055406 | PGDB_C004695 | PGDB_AS000571 | View | |
| IC50 | - | < | 1 | nM | - | — | - | - | MV-4-11 | WO2022073469A1 | PGDB_A069413 | PGDB_C004695 | PGDB_AS000477 | View | |
| IC50 | - | < | 10 | nM | - | — | - | - | MV-4-11 | WO2022073469A1 | PGDB_A077675 | PGDB_C004695 | PGDB_AS002199 | View |