Activity record

PGDB_A021463

Assay: % DegradationTarget: CSNK1A1QC: ambiguous
Activity overview

degradation = 33.2 %

TargetCSNK1A1
Concentration100 nM
Assay / Readout% Degradation
Assay IDPGDB_AS000209
PatentWO2024059107A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C002820
Compound IDPGDB_C002820
Compound72;72;72
Source record IDPGDB_C002820
InChIKeyBUKXXJVKMXZXHH-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000209
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Concentration100 nM
Detection targetprotein_degradation
TargetCSNK1A1
E3Not specified

Source evidence

Patent IDWO2024059107A1
Compound location

72;72;72

72;72;72 enlarged structure72;72;72 location on patent page 10
Activity table
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