Activity record

PGDB_A026371

Assay: viabilityQC: ambiguous
Activity overview

IC50 = 1000-2000 nM

Cell lineTHP-1
Assay / ReadoutIC50 / viability
Assay IDPGDB_AS000638
PatentCN117756818A
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C000379
Compound IDPGDB_C000379
CompounddBET6
Source record IDPGDB_C000379
InChIKeyJGQPZPLJOBHHBK-UFXYQILXSA-N

Assay context

Assay IDPGDB_AS000638
Assay familyviability
Assay systemcell_based
ReadoutIC50
TargetBRD4
E3Not specified
Cell lineTHP-1

Source evidence

Patent IDCN117756818A
Compound location

dBET6

dBET6 enlarged structuredBET6 location on patent page 18
Activity table
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