Assay

PGDB_AS000638

System: cell_basedTarget: BRD4Cell line: THP-1
Assay context summary

Assay context

22 activity records
Assay familyviability
Systemcell_based
ReadoutIC50
TargetBRD4
E3Not specified
Cell lineTHP-1
Activity compounds and values

Activity records

22 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C000363
IC50-=100-1000nM-—--THP-1CN117756818APGDB_A011829PGDB_C000363PGDB_AS000638View
2D structure for PGDB_C000365
IC50-<100nM-—--THP-1CN117756818APGDB_A014202PGDB_C000365PGDB_AS000638View
2D structure for PGDB_C000360
IC50-=100-1000nM-—--THP-1CN117756818APGDB_A015433PGDB_C000360PGDB_AS000638View
2D structure for PGDB_C000371
IC50-<100nM-—--THP-1CN117756818APGDB_A018003PGDB_C000371PGDB_AS000638View
2D structure for PGDB_C000373
IC50-=17.9nM-—--THP-1CN117756818APGDB_A021808PGDB_C000373PGDB_AS000638View
2D structure for PGDB_C000366
IC50-<100nM-—--THP-1CN117756818APGDB_A025624PGDB_C000366PGDB_AS000638View
2D structure for PGDB_C000367
IC50-<100nM-—--THP-1CN117756818APGDB_A026332PGDB_C000367PGDB_AS000638View
2D structure for PGDB_C000379
IC50-=1000-2000nM-—--THP-1CN117756818APGDB_A026371PGDB_C000379PGDB_AS000638View
2D structure for PGDB_C000059
IC50->2000nM-—--THP-1CN117756818APGDB_A026786PGDB_C000059PGDB_AS000638View
2D structure for PGDB_C000362
IC50-=100-1000nM-—--THP-1CN117756818APGDB_A034342PGDB_C000362PGDB_AS000638View
2D structure for PGDB_C000361
IC50-=100-1000nM-—--THP-1CN117756818APGDB_A041347PGDB_C000361PGDB_AS000638View
2D structure for PGDB_C000378
IC50->2000nM-—--THP-1CN117756818APGDB_A042421PGDB_C000378PGDB_AS000638View
2D structure for PGDB_C000376
IC50-<100nM-—--THP-1CN117756818APGDB_A043326PGDB_C000376PGDB_AS000638View
2D structure for PGDB_C000374
IC50-=16.44nM-—--THP-1CN117756818APGDB_A046241PGDB_C000374PGDB_AS000638View
2D structure for PGDB_C000375
IC50-<100nM-—--THP-1CN117756818APGDB_A050552PGDB_C000375PGDB_AS000638View
2D structure for PGDB_C000368
IC50-<100nM-—--THP-1CN117756818APGDB_A053452PGDB_C000368PGDB_AS000638View
2D structure for PGDB_C000364
IC50-=102.7nM-—--THP-1CN117756818APGDB_A056478PGDB_C000364PGDB_AS000638View
2D structure for PGDB_C000359
IC50-=100-1000nM-—--THP-1CN117756818APGDB_A060541PGDB_C000359PGDB_AS000638View
2D structure for PGDB_C000372
IC50-=31.96nM-—--THP-1CN117756818APGDB_A061716PGDB_C000372PGDB_AS000638View
2D structure for PGDB_C000377
IC50->2000nM-—--THP-1CN117756818APGDB_A061893PGDB_C000377PGDB_AS000638View
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