Activity record

PGDB_A028785

Assay: % DegradationTarget: GSPT1QC: ambiguous
Activity overview

degradation = 11.1 %

TargetGSPT1
Concentration1 uM
Assay / Readout% Degradation
Assay IDPGDB_AS001974
PatentWO2024059107A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C002809
Compound IDPGDB_C002809
Compound56;56;56
Source record IDPGDB_C002809
InChIKeyVWGBLNAJOOBMEC-UXBLZVDNSA-N

Assay context

Assay IDPGDB_AS001974
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Concentration1 uM
Detection targetprotein_degradation
TargetGSPT1
E3Not specified

Source evidence

Patent IDWO2024059107A1
Compound location

56;56;56

56;56;56 enlarged structure56;56;56 location on patent page 9
Activity table
Page 141 · table single