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Compound
PGDB_C002809
8 activity records1 related patents
2D structure
O=C(/C=C/c1ccccc1)Nc1ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=OCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 60.2 | % | 100 nM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A020835 | PGDB_C002809 | PGDB_AS000209 | View |
| % Degradation | - | = | 67 | % | 1 uM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A025242 | PGDB_C002809 | PGDB_AS000685 | View |
| % Degradation | - | = | 7.6 | % | 100 nM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A026116 | PGDB_C002809 | PGDB_AS002431 | View |
| % Degradation | - | = | 11.1 | % | 1 uM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A028785 | PGDB_C002809 | PGDB_AS001974 | View |
| % Degradation | - | = | 70.8 | % | 100 nM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A050381 | PGDB_C002809 | PGDB_AS001414 | View |
| % Degradation | - | = | 13.1 | % | 100 nM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A054940 | PGDB_C002809 | PGDB_AS000707 | View |
| % Degradation | - | = | 29.4 | % | 1 uM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A071366 | PGDB_C002809 | PGDB_AS000768 | View |
| % Degradation | - | = | 89.6 | % | 1 uM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A074341 | PGDB_C002809 | PGDB_AS000892 | View |