Activity record

PGDB_A030040

Assay: biochemicalTarget: CRBNQC: standardized
Activity overview

IC50 = 27 nM

TargetCRBN
E3 ligaseCRBN
Time3 h
Assay / ReadoutHTRF / IC50
Assay IDPGDB_AS001113
PatentCA3286762A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C021277
Compound IDPGDB_C021277
CompoundExample 30
Source record IDPGDB_C021277
InChIKeyDMOOHDDOAZYPDX-NDEPHWFRSA-N

Assay context

Assay IDPGDB_AS001113
Assay familybiochemical
Assay systembiochemical
ReadoutIC50
TechnologyHTRF
Treatment time3 h
TargetCRBN
E3CRBN

Source evidence

Patent IDCA3286762A1
Compound location

Example 30

Example 30 enlarged structureExample 30 location on patent page 78
Activity table
Page 103 · table single