Assay
PGDB_AS001113
System: biochemicalTarget: CRBN
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 38 | nM | - | — | CRBN | CRBN | - | CA3286762A1 | PGDB_A019449 | PGDB_C025619 | PGDB_AS001113 | View | |
| IC50 | - | = | 20 | nM | - | — | CRBN | CRBN | - | CA3286762A1 | PGDB_A019599 | PGDB_C025616 | PGDB_AS001113 | View | |
| IC50 | - | = | 27 | nM | - | — | CRBN | CRBN | - | CA3286762A1 | PGDB_A030040 | PGDB_C021277 | PGDB_AS001113 | View | |
| IC50 | - | = | 8 | nM | - | — | CRBN | CRBN | - | CA3286762A1 | PGDB_A054030 | PGDB_C025631 | PGDB_AS001113 | View | |
| IC50 | - | = | 19 | nM | - | — | CRBN | CRBN | - | CA3286762A1 | PGDB_A075271 | PGDB_C025617 | PGDB_AS001113 | View | |
| IC50 | - | = | 34 | nM | - | — | CRBN | CRBN | - | CA3286762A1 | PGDB_A075299 | PGDB_C025615 | PGDB_AS001113 | View |