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SIMM · NJU

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A patent-derived molecular glue bioactivity database with traceable evidence.

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SIMM · NJU

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SIMM · NJU

Activity record

PGDB_A037219

Assay: viabilityTarget: BTKQC: ambiguous

Activity overview

IC50 < 50 nM

TargetBTK

E3 ligaseCRBN

Cell line22Rv1

Time96 h

Assay / ReadoutCCK-8 / viability

Assay IDPGDB_AS001253

PatentCN116239566A

QC statusambiguous

Evidence details

Compound, assay context, and source

Compound

Compound IDPGDB_C019593

CompoundGT-03264

Source record IDPGDB_C019593

InChIKeyHSTNZJQZESPLGQ-ASYYUYISSA-N

Assay context

Assay IDPGDB_AS001253

Assay familyviability

Assay systemcell_based

Readoutviability

TechnologyCCK-8

Treatment time96 h

Detection target% Cell viability

TargetBTK

E3CRBN

Cell line22Rv1

OrganismHomo sapiens

Source evidence

Patent IDCN116239566A

Compound location

GT-03264

GT-03264 enlarged structure

GT-03264 location on patent page 278

Activity table

Page 844 · table start

Page 845 · table end

A patent-derived molecular glue bioactivity database with traceable evidence.

Global reach

0

0 countries/regions

·

SIMM · NJU