Assay
PGDB_AS001253
System: cell_basedCell line: 22Rv1
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | BTK | CRBN | 22Rv1 | CN116239566A | PGDB_A014476 | PGDB_C025809 | PGDB_AS001253 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | CRBN | 22Rv1 | CN116239566A | PGDB_A024066 | PGDB_C025808 | PGDB_AS001253 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | CRBN | 22Rv1 | CN116239566A | PGDB_A037219 | PGDB_C019593 | PGDB_AS001253 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | CRBN | 22Rv1 | CN116239566A | PGDB_A038115 | PGDB_C015982 | PGDB_AS001253 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | CRBN | 22Rv1 | CN116239566A | PGDB_A041982 | PGDB_C025815 | PGDB_AS001253 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | CRBN | 22Rv1 | CN116239566A | PGDB_A058104 | PGDB_C025807 | PGDB_AS001253 | View |