Activity record

PGDB_A041308

Assay: % DegradationTarget: CSNK1A1QC: ambiguous
Activity overview

degradation = 64 %

TargetCSNK1A1
Concentration1 uM
Assay / Readout% Degradation
Assay IDPGDB_AS000685
PatentWO2024059107A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C002828
Compound IDPGDB_C002828
Compound75;75
Source record IDPGDB_C002828
InChIKeySSGXQMNAQRSFRQ-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000685
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Concentration1 uM
Detection targetprotein_degradation
TargetCSNK1A1
E3Not specified

Source evidence

Patent IDWO2024059107A1
Compound location

75;75

75;75 enlarged structure75;75 location on patent page 94
Activity table
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