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Compound
PGDB_C002828
8 activity records1 related patents
2D structure
COc1cc(Oc2ccccc2)ccc1C(=O)Nc1ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=OCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 7 | % | 1 uM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A008146 | PGDB_C002828 | PGDB_AS000768 | View |
| % Degradation | - | = | 48.1 | % | 100 nM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A009504 | PGDB_C002828 | PGDB_AS000209 | View |
| % Degradation | - | = | 2.4 | % | 100 nM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A013018 | PGDB_C002828 | PGDB_AS000707 | View |
| % Degradation | - | = | 12.6 | % | 1 uM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A034864 | PGDB_C002828 | PGDB_AS001974 | View |
| % Degradation | - | = | 83.3 | % | 1 uM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A038952 | PGDB_C002828 | PGDB_AS000892 | View |
| % Degradation | - | = | 0.4 | % | 100 nM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A039376 | PGDB_C002828 | PGDB_AS002431 | View |
| % Degradation | - | = | 64 | % | 1 uM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A041308 | PGDB_C002828 | PGDB_AS000685 | View |
| % Degradation | - | = | 54.6 | % | 100 nM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A049098 | PGDB_C002828 | PGDB_AS001414 | View |