Activity record

PGDB_A051861

Assay: biochemicalTarget: CDK12QC: ambiguous
Activity overview

IC50 = 21 nM

TargetCDK12
Time60 min
Assay / ReadoutIC50 / biochemical
Assay IDPGDB_AS001066
PatentCN114929708B
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006610
Compound IDPGDB_C006610
CompoundH-APPAMP-043;H-APPAMP-043
Source record IDPGDB_C006610
InChIKeyZRVMIIBSDSMIEO-XLIONFOSSA-N

Assay context

Assay IDPGDB_AS001066
Assay familybiochemical
Assay systembiochemical
ReadoutIC50
Treatment time60 min
TargetCDK12
E3Not specified
OrganismHomo sapiens

Source evidence

Patent IDCN114929708B
Compound location

H-APPAMP-043;H-APPAMP-043

H-APPAMP-043;H-APPAMP-043 enlarged structureH-APPAMP-043;H-APPAMP-043 location on patent page 47
Activity table
Page 197 · table single