Activity record

PGDB_A057550

Assay: biochemicalTarget: CDK7QC: ambiguous
Activity overview

IC50 = 274 nM

TargetCDK7
Time60 min
Assay / ReadoutIC50 / biochemical
Assay IDPGDB_AS002150
PatentCN114929708B
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006597
Compound IDPGDB_C006597
CompoundH-APPAMP-030
Source record IDPGDB_C006597
InChIKeyOFFUMIIHKYXTSP-GCJKJVERSA-N

Assay context

Assay IDPGDB_AS002150
Assay familybiochemical
Assay systembiochemical
ReadoutIC50
Treatment time60 min
TargetCDK7
E3Not specified
OrganismHomo sapiens

Source evidence

Patent IDCN114929708B
Compound location

H-APPAMP-030

H-APPAMP-030 enlarged structureH-APPAMP-030 location on patent page 43
Activity table
Page 195 · table start
Page 196 · table middle
Page 197 · table end