Assay context summary

Assay context

48 activity records
Activity compounds and values

Activity records

48 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C006600
IC50-=1060nM-CDK7--CN114929708BPGDB_A009300PGDB_C006600PGDB_AS002150View
2D structure for PGDB_C006571
IC50-=305nM-CDK7--CN114929708BPGDB_A012717PGDB_C006571PGDB_AS002150View
2D structure for PGDB_C006578
IC50-=168nM-CDK7--CN114929708BPGDB_A013923PGDB_C006578PGDB_AS002150View
2D structure for PGDB_C006581
IC50-=19nM-CDK7--CN114929708BPGDB_A015574PGDB_C006581PGDB_AS002150View
2D structure for PGDB_C006599
IC50-=859nM-CDK7--CN114929708BPGDB_A018948PGDB_C006599PGDB_AS002150View
2D structure for PGDB_C006582
IC50-=3nM-CDK7--CN114929708BPGDB_A019504PGDB_C006582PGDB_AS002150View
2D structure for PGDB_C006601
IC50-=152nM-CDK7--CN114929708BPGDB_A019615PGDB_C006601PGDB_AS002150View
2D structure for PGDB_C006585
IC50-=206nM-CDK7--CN114929708BPGDB_A019767PGDB_C006585PGDB_AS002150View
2D structure for PGDB_C006577
IC50-=238nM-CDK7--CN114929708BPGDB_A019852PGDB_C006577PGDB_AS002150View
2D structure for PGDB_C006588
IC50-=28nM-CDK7--CN114929708BPGDB_A023093PGDB_C006588PGDB_AS002150View
2D structure for PGDB_C006569
IC50-=704nM-CDK7--CN114929708BPGDB_A023581PGDB_C006569PGDB_AS002150View
2D structure for PGDB_C006570
IC50-=411nM-CDK7--CN114929708BPGDB_A023749PGDB_C006570PGDB_AS002150View
2D structure for PGDB_C006579
IC50-=214nM-CDK7--CN114929708BPGDB_A029805PGDB_C006579PGDB_AS002150View
2D structure for PGDB_C006580
IC50-=226nM-CDK7--CN114929708BPGDB_A032463PGDB_C006580PGDB_AS002150View
2D structure for PGDB_C006592
IC50-=334nM-CDK7--CN114929708BPGDB_A032524PGDB_C006592PGDB_AS002150View
2D structure for PGDB_C006596
IC50-=196nM-CDK7--CN114929708BPGDB_A034822PGDB_C006596PGDB_AS002150View
2D structure for PGDB_C006589
IC50-=622nM-CDK7--CN114929708BPGDB_A037393PGDB_C006589PGDB_AS002150View
2D structure for PGDB_C006603
IC50-=1150nM-CDK7--CN114929708BPGDB_A039019PGDB_C006603PGDB_AS002150View
2D structure for PGDB_C006605
IC50-=762nM-CDK7--CN114929708BPGDB_A042047PGDB_C006605PGDB_AS002150View
2D structure for PGDB_C006609
IC50-=974nM-CDK7--CN114929708BPGDB_A044619PGDB_C006609PGDB_AS002150View