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SIMM · NJU
Assay
PGDB_AS002150
System: biochemical
Target: CDK7
Assay context summary
Assay context
48 activity records
Assay family
biochemical
System
biochemical
Readout
IC50
Target
CDK7
E3
Not specified
Organism
Homo sapiens
Activity compounds and values
Activity records
48 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
IC50
-
=
1060
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A009300
PGDB_C006600
PGDB_AS002150
View
IC50
-
=
305
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A012717
PGDB_C006571
PGDB_AS002150
View
IC50
-
=
168
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A013923
PGDB_C006578
PGDB_AS002150
View
IC50
-
=
19
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A015574
PGDB_C006581
PGDB_AS002150
View
IC50
-
=
859
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A018948
PGDB_C006599
PGDB_AS002150
View
IC50
-
=
3
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A019504
PGDB_C006582
PGDB_AS002150
View
IC50
-
=
152
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A019615
PGDB_C006601
PGDB_AS002150
View
IC50
-
=
206
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A019767
PGDB_C006585
PGDB_AS002150
View
IC50
-
=
238
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A019852
PGDB_C006577
PGDB_AS002150
View
IC50
-
=
28
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A023093
PGDB_C006588
PGDB_AS002150
View
IC50
-
=
704
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A023581
PGDB_C006569
PGDB_AS002150
View
IC50
-
=
411
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A023749
PGDB_C006570
PGDB_AS002150
View
IC50
-
=
214
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A029805
PGDB_C006579
PGDB_AS002150
View
IC50
-
=
226
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A032463
PGDB_C006580
PGDB_AS002150
View
IC50
-
=
334
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A032524
PGDB_C006592
PGDB_AS002150
View
IC50
-
=
196
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A034822
PGDB_C006596
PGDB_AS002150
View
IC50
-
=
622
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A037393
PGDB_C006589
PGDB_AS002150
View
IC50
-
=
1150
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A039019
PGDB_C006603
PGDB_AS002150
View
IC50
-
=
762
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A042047
PGDB_C006605
PGDB_AS002150
View
IC50
-
=
974
nM
-
—
CDK7
-
-
CN114929708B
PGDB_A044619
PGDB_C006609
PGDB_AS002150
View