Activity record

PGDB_A059276

Assay: % DegradationTarget: GSPT1QC: ambiguous
Activity overview

degradation = 30-60 %

TargetGSPT1
Concentration1 uM
Assay / Readout% Degradation
Assay IDPGDB_AS001783
PatentCN117683022A
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C000344
Compound IDPGDB_C000344
Compound6;6
Source record IDPGDB_C000344
InChIKeyZEVWOCAIKRDLAT-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001783
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Concentration1 uM
Detection targetprotein_degradation
TargetGSPT1
E3Not specified

Source evidence

Patent IDCN117683022A
Compound location

6;6

6;6 enlarged structure6;6 location on patent page 3
Activity table
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