Activity record

PGDB_A068294

Assay: biochemicalQC: ambiguous
Activity overview

selectivity_index = 1.9 fold

Time60 min
ControlCDK7 / CDK12
Assay / ReadoutFold change / biochemical
Assay IDPGDB_AS002236
PatentCN114929708B
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006583
Compound IDPGDB_C006583
CompoundH-APPAMP-016;H-APPAMP-016
Source record IDPGDB_C006583
InChIKeyKLPZXNIXEQAIRZ-APWZRJJASA-N

Assay context

Assay IDPGDB_AS002236
Assay familybiochemical
Assay systembiochemical
ReadoutFold change
Treatment time60 min
TargetCDK12 | CDK7
E3Not specified
OrganismHomo sapiens

Source evidence

Patent IDCN114929708B
Compound location

H-APPAMP-016;H-APPAMP-016

H-APPAMP-016;H-APPAMP-016 enlarged structureH-APPAMP-016;H-APPAMP-016 location on patent page 40
Activity table
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