Activity record

PGDB_A072641

Assay: biochemicalTarget: CDK12QC: ambiguous
Activity overview

IC50 = 540 nM

TargetCDK12
Time60 min
Assay / ReadoutIC50 / biochemical
Assay IDPGDB_AS001268
PatentCN114929708B
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006587
Compound IDPGDB_C006587
CompoundH-APPAMP-020;H-APPAMP-020
Source record IDPGDB_C006587
InChIKeyMHHLCQCUGOXPSF-XLIONFOSSA-N

Assay context

Assay IDPGDB_AS001268
Assay familybiochemical
Assay systembiochemical
ReadoutIC50
Treatment time60 min
TargetCDK12
E3Not specified
OrganismHomo sapiens

Source evidence

Patent IDCN114929708B
Compound location

H-APPAMP-020;H-APPAMP-020

H-APPAMP-020;H-APPAMP-020 enlarged structureH-APPAMP-020;H-APPAMP-020 location on patent page 41
Activity table
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