Activity record

PGDB_A072887

Assay: % DegradationTarget: GSPT1QC: standardized
Activity overview

DC50 = 34.16 nM

TargetGSPT1
Cell lineU937
Time6 h
Assay / ReadoutWestern_blot / DC50
Assay IDPGDB_AS002566
PatentCN117917402A
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C000496
Compound IDPGDB_C000496
CompoundWYY-26
Source record IDPGDB_C000530
InChIKeyQCCCAEGSQRBURI-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS002566
Assay family% Degradation
Assay systemcell_based
ReadoutDC50
TechnologyWestern_blot
Treatment time6 h
TargetGSPT1
E3Not specified
Cell lineU937

Source evidence

Patent IDCN117917402A
Activity table
Page 48 · table start
Page 49 · table end