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O=C1CCC(N2Cc3ccc(CCC(=O)Nc4ccc(-c5ccc(C(F)(F)F)cc5)c(CN5CCOCC5)c4)cc3C2=O)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 9.611 | nM | - | — | GSPT1 | - | MV-4-11 | CN117917402A | PGDB_A013454 | PGDB_C000496 | PGDB_AS000703 | View | |
| IC50 | - | = | 27.2 | nM | - | — | GSPT1 | - | U937 | CN117917402A | PGDB_A015483 | PGDB_C000496 | PGDB_AS002565 | View | |
| IC50 | - | = | 771.1 | nM | - | — | GSPT1 | - | H1299 | CN117917402A | PGDB_A044241 | PGDB_C000496 | PGDB_AS002493 | View | |
| IC50 | - | = | 40.67 | nM | - | — | - | - | MOLT-4 | CN117917402A | PGDB_A071939 | PGDB_C000496 | PGDB_AS002289 | View | |
| DC50 | - | = | 34.16 | nM | - | — | GSPT1 | - | U937 | CN117917402A | PGDB_A072887 | PGDB_C000496 | PGDB_AS002566 | View |