Assay

PGDB_AS002566

System: cell_basedTarget: GSPT1Cell line: U937
Assay context summary

Assay context

34 activity records
Assay family% Degradation
Systemcell_based
ReadoutDC50
TargetGSPT1
E3Not specified
Cell lineU937
TechnologyWestern_blot
Activity compounds and values

Activity records

34 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C000498
DC50-=702.1nM-—GSPT1-U937CN117917402APGDB_A007093PGDB_C000498PGDB_AS002566View
2D structure for PGDB_C000487
DC50-=86.4nM-—GSPT1-U937CN117917402APGDB_A009268PGDB_C000487PGDB_AS002566View
2D structure for PGDB_C000494
DC50-=283.4nM-—GSPT1-U937CN117917402APGDB_A012736PGDB_C000494PGDB_AS002566View
2D structure for PGDB_C000476
DC50->10000nM-—GSPT1-U937CN117917402APGDB_A013841PGDB_C000476PGDB_AS002566View
2D structure for PGDB_C000493
DC50-=212.4nM-—GSPT1-U937CN117917402APGDB_A016636PGDB_C000493PGDB_AS002566View
2D structure for PGDB_C000485
DC50-=176.3nM-—GSPT1-U937CN117917402APGDB_A020628PGDB_C000485PGDB_AS002566View
2D structure for PGDB_C000477
DC50-=3858nM-—GSPT1-U937CN117917402APGDB_A020815PGDB_C000477PGDB_AS002566View
2D structure for PGDB_C000478
DC50-=447.2nM-—GSPT1-U937CN117917402APGDB_A021334PGDB_C000478PGDB_AS002566View
2D structure for PGDB_C000503
DC50->10000nM-—GSPT1-U937CN117917402APGDB_A024843PGDB_C000503PGDB_AS002566View
2D structure for PGDB_C000486
DC50-=35nM-—GSPT1-U937CN117917402APGDB_A025494PGDB_C000486PGDB_AS002566View
2D structure for PGDB_C000479
DC50->10000nM-—GSPT1-U937CN117917402APGDB_A029181PGDB_C000479PGDB_AS002566View
2D structure for PGDB_C000484
DC50-=2204nM-—GSPT1-U937CN117917402APGDB_A030783PGDB_C000484PGDB_AS002566View
2D structure for PGDB_C000483
DC50->10000nM-—GSPT1-U937CN117917402APGDB_A034118PGDB_C000483PGDB_AS002566View
2D structure for PGDB_C000482
DC50->10000nM-—GSPT1-U937CN117917402APGDB_A035249PGDB_C000482PGDB_AS002566View
2D structure for PGDB_C000475
DC50-=373.8nM-—GSPT1-U937CN117917402APGDB_A036046PGDB_C000475PGDB_AS002566View
2D structure for PGDB_C000488
DC50-=220.6nM-—GSPT1-U937CN117917402APGDB_A037809PGDB_C000488PGDB_AS002566View
2D structure for PGDB_C000497
DC50-=11.8nM-—GSPT1-U937CN117917402APGDB_A038248PGDB_C000497PGDB_AS002566View
2D structure for PGDB_C000502
DC50-=37.45nM-—GSPT1-U937CN117917402APGDB_A038585PGDB_C000502PGDB_AS002566View
2D structure for PGDB_C000490
DC50-=251.1nM-—GSPT1-U937CN117917402APGDB_A041047PGDB_C000490PGDB_AS002566View
2D structure for PGDB_C000504
DC50->10000nM-—GSPT1-U937CN117917402APGDB_A041175PGDB_C000504PGDB_AS002566View
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