Activity record

PGDB_A078479

Assay: % DegradationTarget: VAV1QC: ambiguous
Activity overview

DC50 <= 20 nM

TargetVAV1
Cell lineprimary_human_blood
Assay / ReadoutDC50 / % Degradation
Assay IDPGDB_AS001692
PatentWO2026114367A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C029566
Compound IDPGDB_C029566
Compound化合物 9
Source record IDPGDB_C029566
InChIKeyCXFYGRLONQOGHW-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001692
Assay family% Degradation
Assay systemcell_based
ReadoutDC50
TargetVAV1
E3Not specified
Cell lineprimary_human_blood
OrganismHomo sapiens

Source evidence

Patent IDWO2026114367A1
Compound location

化合物 9

化合物 9 enlarged structure化合物 9 location on patent page 88
Activity table
Page 204 · table start
Page 205 · table end