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Compound
PGDB_C029566
7 activity records2 related patents
2D structure
O=C1CCC(c2cccc(-c3ccc(-n4cccc(OC5CC5)c4=O)cc3)c2Cl)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | <= | 1 | nM | - | — | VAV1 | - | primaryT | WO2026114367A1 | PGDB_A000754 | PGDB_C029566 | PGDB_AS000152 | View |
| DC50 | - | <= | 20 | nM | - | — | VAV1 | - | - | WO2026114367A1 | PGDB_A003936 | PGDB_C029566 | PGDB_AS000190 | View |
| IC50 | - | <= | 1 | nM | - | — | VAV1 | - | primaryT | WO2026114367A1 | PGDB_A005377 | PGDB_C029566 | PGDB_AS002534 | View |
| DC50 | - | = | 2.3 | nM | - | — | VAV1 | - | - | WO2026051943A1 | PGDB_A006231 | PGDB_C029566 | PGDB_AS001440 | View |
| DC50 | - | <= | 20 | nM | - | — | VAV1 | - | primary_human_blood | WO2026114367A1 | PGDB_A078479 | PGDB_C029566 | PGDB_AS001692 | View |
| Dmax | - | = | 98.8 | % | Concentration series: 10 uM, 1 uM | - | VAV1 | - | - | WO2026051943A1 | PGDB_A080915 | PGDB_C029566 | PGDB_AS000777 | View |
| IC50 | - | <= | 1 | nM | - | — | VAV1 | - | primary T cells | WO2026114367A1 | PGDB_A081767 | PGDB_C029566 | PGDB_AS000754 | View |