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SIMM · NJU
Assay
PGDB_AS001692
System: cell_based
Target: VAV1
Cell line: primary_human_blood
Assay context summary
Assay context
63 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
VAV1
E3
Not specified
Cell line
primary_human_blood
Organism
Homo sapiens
Activity compounds and values
Activity records
63 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A000384
PGDB_C031733
PGDB_AS001692
View
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A000420
PGDB_C031687
PGDB_AS001692
View
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A000462
PGDB_C031702
PGDB_AS001692
View
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A000545
PGDB_C031686
PGDB_AS001692
View
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A000583
PGDB_C031740
PGDB_AS001692
View
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A001008
PGDB_C031721
PGDB_AS001692
View
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A001263
PGDB_C031704
PGDB_AS001692
View
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A001304
PGDB_C031717
PGDB_AS001692
View
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A001453
PGDB_C031684
PGDB_AS001692
View
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A001505
PGDB_C031682
PGDB_AS001692
View
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A001652
PGDB_C031725
PGDB_AS001692
View
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A001708
PGDB_C031732
PGDB_AS001692
View
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A002059
PGDB_C031736
PGDB_AS001692
View
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A002195
PGDB_C031688
PGDB_AS001692
View
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A002457
PGDB_C031694
PGDB_AS001692
View
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A002653
PGDB_C031728
PGDB_AS001692
View
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A002691
PGDB_C031696
PGDB_AS001692
View
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A002910
PGDB_C031711
PGDB_AS001692
View
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A002938
PGDB_C031723
PGDB_AS001692
View
DC50
-
<=
20
nM
-
—
VAV1
-
primary_human_blood
WO2026114367A1
PGDB_A003073
PGDB_C031718
PGDB_AS001692
View