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SIMM · NJU
Assay
PGDB_AS000025
System: cell_based
Cell line: HEK293
Assay context summary
Assay context
87 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
E3
Not specified
Cell line
HEK293
Activity compounds and values
Activity records
87 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
13
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A007619
PGDB_C008075
PGDB_AS000025
View
Dmax
-
=
17
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A008747
PGDB_C008095
PGDB_AS000025
View
Dmax
-
=
17
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A009048
PGDB_C008067
PGDB_AS000025
View
Dmax
-
=
11
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A010076
PGDB_C008060
PGDB_AS000025
View
Dmax
-
=
0.75
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A011047
PGDB_C008064
PGDB_AS000025
View
Dmax
-
=
14
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A011175
PGDB_C008083
PGDB_AS000025
View
Dmax
-
=
0.35
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A011430
PGDB_C008120
PGDB_AS000025
View
Dmax
-
=
0.84
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A014501
PGDB_C008076
PGDB_AS000025
View
Dmax
-
=
4.3
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A014856
PGDB_C008125
PGDB_AS000025
View
Dmax
-
=
0.2
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A015672
PGDB_C008066
PGDB_AS000025
View
Dmax
-
=
6.1
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A016234
PGDB_C008104
PGDB_AS000025
View
Dmax
-
=
2
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A016408
PGDB_C008053
PGDB_AS000025
View
Dmax
-
=
14
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A016941
PGDB_C008046
PGDB_AS000025
View
Dmax
-
=
1.5
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A019678
PGDB_C008093
PGDB_AS000025
View
Dmax
-
=
0.16
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A020995
PGDB_C008132
PGDB_AS000025
View
Dmax
-
=
0.51
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A023272
PGDB_C008073
PGDB_AS000025
View
Dmax
-
=
3.5
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A023643
PGDB_C008072
PGDB_AS000025
View
Dmax
-
=
14
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A025436
PGDB_C008056
PGDB_AS000025
View
Dmax
-
=
8.4
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A025952
PGDB_C008096
PGDB_AS000025
View
Dmax
-
=
10
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A026134
PGDB_C008081
PGDB_AS000025
View