Assay context summary

Assay context

169 activity records
Activity compounds and values

Activity records

169 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C029568
IC50-=0.034nM-VAV1-pan-TWO2026051943A1PGDB_A000131PGDB_C029568PGDB_AS000112View
2D structure for PGDB_C029593
IC50-=0.052nM-VAV1-pan-TWO2026051943A1PGDB_A000163PGDB_C029593PGDB_AS000112View
2D structure for PGDB_C029492
IC50-=0.0091nM-VAV1-pan-TWO2026051943A1PGDB_A000187PGDB_C029492PGDB_AS000112View
2D structure for PGDB_C029477
IC50-=0.23nM-VAV1-pan-TWO2026051943A1PGDB_A000245PGDB_C029477PGDB_AS000112View
2D structure for PGDB_C029565
IC50-=0.074nM-VAV1-pan-TWO2026051943A1PGDB_A000281PGDB_C029565PGDB_AS000112View
2D structure for PGDB_C029485
IC50-=0.048nM-VAV1-pan-TWO2026051943A1PGDB_A000283PGDB_C029485PGDB_AS000112View
2D structure for PGDB_C029544
IC50-=0.043nM-VAV1-pan-TWO2026051943A1PGDB_A000284PGDB_C029544PGDB_AS000112View
2D structure for PGDB_C029597
IC50-=0.067nM-VAV1-pan-TWO2026051943A1PGDB_A000356PGDB_C029597PGDB_AS000112View
2D structure for PGDB_C029479
IC50-=0.43nM-VAV1-pan-TWO2026051943A1PGDB_A000407PGDB_C029479PGDB_AS000112View
2D structure for PGDB_C029586
IC50-=0.1nM-VAV1-pan-TWO2026051943A1PGDB_A000428PGDB_C029586PGDB_AS000112View
2D structure for PGDB_C029524
IC50-=0.035nM-VAV1-pan-TWO2026051943A1PGDB_A000441PGDB_C029524PGDB_AS000112View
2D structure for PGDB_C029558
IC50-=0.066nM-VAV1-pan-TWO2026051943A1PGDB_A000444PGDB_C029558PGDB_AS000112View
2D structure for PGDB_C029527
IC50-=0.11nM-VAV1-pan-TWO2026051943A1PGDB_A000465PGDB_C029527PGDB_AS000112View
2D structure for PGDB_C029532
IC50-=0.49nM-VAV1-pan-TWO2026051943A1PGDB_A000474PGDB_C029532PGDB_AS000112View
2D structure for PGDB_C029532
IC50-=0.49nM-VAV1-pan-TWO2026051943A1PGDB_A000489PGDB_C029532PGDB_AS000112View
2D structure for PGDB_C029583
IC50-=0.053nM-VAV1-pan-TWO2026051943A1PGDB_A000569PGDB_C029583PGDB_AS000112View
2D structure for PGDB_C029588
IC50-=0.049nM-VAV1-pan-TWO2026051943A1PGDB_A000878PGDB_C029588PGDB_AS000112View
2D structure for PGDB_C029514
IC50-=0.041nM-VAV1-pan-TWO2026051943A1PGDB_A000903PGDB_C029514PGDB_AS000112View
2D structure for PGDB_C029686
IC50-=2.11nM-VAV1-pan-TWO2026051943A1PGDB_A000920PGDB_C029686PGDB_AS000112View
2D structure for PGDB_C029689
IC50-=4.64nM-VAV1-pan-TWO2026051943A1PGDB_A001240PGDB_C029689PGDB_AS000112View