Assay

PGDB_AS000153

System: biochemicalTarget: CRBN | DDB1
Assay context summary

Assay context

42 activity records
Assay familybinding
Systembiochemical
ReadoutKi
TargetCRBN | DDB1
E3CRBN | DDB1
Technologyfluorescence
Activity compounds and values

Activity records

42 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C019055
Ki-=1-10uM-—CRBNCRBN-AU2020392427A1PGDB_A007164PGDB_C019055PGDB_AS000153View
2D structure for PGDB_C019045
Ki-=1-10uM-—CRBNCRBN-AU2020392427A1PGDB_A011501PGDB_C019045PGDB_AS000153View
2D structure for PGDB_C019038
Ki-<=1uM-—CRBNCRBN-AU2020392427A1PGDB_A017100PGDB_C019038PGDB_AS000153View
2D structure for PGDB_C019047
Ki-=1-10uM-—CRBNCRBN-AU2020392427A1PGDB_A017416PGDB_C019047PGDB_AS000153View
2D structure for PGDB_C008731
Ki-=1-10uM-—CRBNCRBN-AU2020392427A1PGDB_A018383PGDB_C008731PGDB_AS000153View
2D structure for PGDB_C019039
Ki-=1-10uM-—CRBNCRBN-AU2020392427A1PGDB_A018843PGDB_C019039PGDB_AS000153View
2D structure for PGDB_C019056
Ki-=10-50uM-—CRBNCRBN-AU2020392427A1PGDB_A019498PGDB_C019056PGDB_AS000153View
2D structure for PGDB_C019053
Ki-=1-10uM-—CRBNCRBN-AU2020392427A1PGDB_A019667PGDB_C019053PGDB_AS000153View
2D structure for PGDB_C019036
Ki-=1-10uM-—CRBNCRBN-AU2020392427A1PGDB_A020675PGDB_C019036PGDB_AS000153View
2D structure for PGDB_C019051
Ki-=1-10uM-—CRBNCRBN-AU2020392427A1PGDB_A023471PGDB_C019051PGDB_AS000153View
2D structure for PGDB_C019043
Ki-=10-50uM-—CRBNCRBN-AU2020392427A1PGDB_A023774PGDB_C019043PGDB_AS000153View
2D structure for PGDB_C019062
Ki-<=1uM-—CRBNCRBN-AU2020392427A1PGDB_A024651PGDB_C019062PGDB_AS000153View
2D structure for PGDB_C019035
Ki-<=1uM-—CRBNCRBN-AU2020392427A1PGDB_A027501PGDB_C019035PGDB_AS000153View
2D structure for PGDB_C019031
Ki-=1-10uM-—CRBNCRBN-AU2020392427A1PGDB_A029349PGDB_C019031PGDB_AS000153View
2D structure for PGDB_C019059
Ki-=1-10uM-—CRBNCRBN-AU2020392427A1PGDB_A031988PGDB_C019059PGDB_AS000153View
2D structure for PGDB_C019057
Ki-=1-10uM-—CRBNCRBN-AU2020392427A1PGDB_A032550PGDB_C019057PGDB_AS000153View
2D structure for PGDB_C019023
Ki-<=1uM-—CRBNCRBN-AU2020392427A1PGDB_A033114PGDB_C019023PGDB_AS000153View
2D structure for PGDB_C019049
Ki-=1-10uM-—CRBNCRBN-AU2020392427A1PGDB_A033582PGDB_C019049PGDB_AS000153View
2D structure for PGDB_C019063
Ki-=1-10uM-—CRBNCRBN-AU2020392427A1PGDB_A038653PGDB_C019063PGDB_AS000153View
2D structure for PGDB_C019040
Ki-<=1uM-—CRBNCRBN-AU2020392427A1PGDB_A039014PGDB_C019040PGDB_AS000153View
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